Search on: SAQUINAVIR 
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Descriptor English:   Saquinavir 
Descriptor Spanish:   Saquinavir 
Descriptor Portuguese:   Saquinavir 
Synonyms English:   Invirase
Ro 31-8959
Saquinavir Mesylate
Saquinavir Monomethanesulfonate
Saquinivir
Monomethanesulfonate, Saquinavir
Ro 31 8959
Ro 318959  
Tree Number:   D03.633.100.531.770
D03.633.100.810.900
Definition English:   An HIV protease inhibitor which acts as an analog of an HIV protease cleavage site. It is a highly specific inhibitor of HIV-1 and HIV-2 proteases, and also inhibits CYTOCHROME P-450 CYP3A. 
Pharmacological Action:   Cytochrome P-450 CYP3A Inhibitors
HIV Protease Inhibitors
 
History Note English:   97; was SAQUINAVIR (NM) 1990-96 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AA analogs & derivatives
AN analysis AI antagonists & inhibitors
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification EC economics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PO poisoning RE radiation effects
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UR urine  
Record Number:   32996 
Unique Identifier:   D019258 

Occurrence in VHL:
 

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